ADC TOXICITY ATLAS
Atlas
Payloads and Linkers
Payloads
Targets
Methods
← Payloads & linkers
Linker
Mal-Val-Ala-PAB
Cleavable
CC(NC(=O)C(NC(=O)CCN1C(=O)C=CC1=O)C(C)C)C(=O)Nc1ccc(CO)cc1
Physicochemistry
Properties
MW
444.488
Da
TPSA
144.91
Ų
xLogP
0.078
Formula
C22H28N4O6
Cleavage
Cleavable
Attachment
Cysteine (interchain)
1 agent
ADCs built on this linker
Any-grade
Grade 3+
Agent · target
Ocular
Hepatic
Neutrop.
Thrombo.
Anemia
GI
ILD
Neuro.
HDP-101
TNFRSF17
0
22
56
33
0%
severity
100%
0
Assessed · clear
true 0%
No data
never assessed